Compile Data Set for Download or QSAR
Found 596 from Lund University
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50479287(CHEMBL487686)copy SMILEScopy InChI
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50479291(CHEMBL469477)copy SMILEScopy InChI
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50479296(CHEMBL488283)copy SMILEScopy InChI
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333162(2-(4-Methylphenyl)-9-[2-(3-thienyl)ethyl]-2,6-dihy...)copy SMILEScopy InChI
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038FKPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50479299(CHEMBL487687)copy SMILEScopy InChI
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50185292(6-Benzyl-4-oxo-1,4-dihydroquinoline-3-carboxylic A...)copy SMILEScopy InChI
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50185292(6-Benzyl-4-oxo-1,4-dihydroquinoline-3-carboxylic A...)copy SMILEScopy InChI
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MZ2PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50479285(CHEMBL471551)copy SMILEScopy InChI
Affinity DataKi:  0.380nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50479295(CHEMBL487685)copy SMILEScopy InChI
Affinity DataKi:  0.390nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333160(9-Methyl-2-phenyl-2,6-dihydro[1,2,4]triazolo[4,3-c...)copy SMILEScopy InChI
Affinity DataKi:  0.430nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038FKPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50479293(CHEMBL520411)copy SMILEScopy InChI
Affinity DataKi:  0.510nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50479290(CHEMBL488284)copy SMILEScopy InChI
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333163(2-(4-Methylphenyl)-9-[2-(3-pyridyl)ethyl]-2,6-dihy...)copy SMILEScopy InChI
Affinity DataKi:  0.680nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038FKPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333162(2-(4-Methylphenyl)-9-[2-(3-thienyl)ethyl]-2,6-dihy...)copy SMILEScopy InChI
Affinity DataKi:  0.710nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha3beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038FKPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Lund University

Curated by ChEMBL
LigandPNGBDBM50293263(2-(5-benzyl-2-hydroxyphenyl)-6-methyl-4H-chromen-4...)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha1beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9Q3ZPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50479294(CHEMBL487688)copy SMILEScopy InChI
Affinity DataKi:  0.880nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50479292(CHEMBL470283)copy SMILEScopy InChI
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333160(9-Methyl-2-phenyl-2,6-dihydro[1,2,4]triazolo[4,3-c...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha2beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038FKPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Lund University

Curated by ChEMBL
LigandPNGBDBM50293262(2-(5-benzyl-2-hydroxyphenyl)-6-methylquinolin-4(1H...)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha1beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9Q3ZPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333160(9-Methyl-2-phenyl-2,6-dihydro[1,2,4]triazolo[4,3-c...)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha3beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038FKPubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333162(2-(4-Methylphenyl)-9-[2-(3-thienyl)ethyl]-2,6-dihy...)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha2beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038FKPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333163(2-(4-Methylphenyl)-9-[2-(3-pyridyl)ethyl]-2,6-dihy...)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha3beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038FKPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(RAT)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293263(2-(5-benzyl-2-hydroxyphenyl)-6-methyl-4H-chromen-4...)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha5beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9Q3ZPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50479288(CHEMBL488286)copy SMILEScopy InChI
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50479289(CHEMBL488285)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333161(2-(4-Methylphenyl)-9-(2-phenylethyl)-2,6-dihydro[1...)copy SMILEScopy InChI
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038FKPubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333162(2-(4-Methylphenyl)-9-[2-(3-thienyl)ethyl]-2,6-dihy...)copy SMILEScopy InChI
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha5beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038FKPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50185296(6-ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone | C...)copy SMILEScopy InChI
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MZ2PubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333163(2-(4-Methylphenyl)-9-[2-(3-pyridyl)ethyl]-2,6-dihy...)copy SMILEScopy InChI
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha2beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038FKPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50479297(CHEMBL506314)copy SMILEScopy InChI
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50479298(CHEMBL206540 | GNF-Pf-4421 | MMV007116)copy SMILEScopy InChI
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50185292(6-Benzyl-4-oxo-1,4-dihydroquinoline-3-carboxylic A...)copy SMILEScopy InChI
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha3 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MZ2PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-5(RAT)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293262(2-(5-benzyl-2-hydroxyphenyl)-6-methylquinolin-4(1H...)copy SMILEScopy InChI
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha5beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9Q3ZPubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333163(2-(4-Methylphenyl)-9-[2-(3-pyridyl)ethyl]-2,6-dihy...)copy SMILEScopy InChI
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha5beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038FKPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333161(2-(4-Methylphenyl)-9-(2-phenylethyl)-2,6-dihydro[1...)copy SMILEScopy InChI
Affinity DataKi:  9.70nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha3beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038FKPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(RAT)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293263(2-(5-benzyl-2-hydroxyphenyl)-6-methyl-4H-chromen-4...)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha3beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9Q3ZPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50479286(CHEMBL487867)copy SMILEScopy InChI
Affinity DataKi:  11nMAssay Description:Displacement of [3H]flumazenil from human recombinant GABAA alpha-1-beta-2-gamma-2S receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0QGQPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50185293(6-bromo-3-ethoxycarbonyl-4-quinolone | CHEMBL20525...)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MZ2PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)copy SMILEScopy InChI
Affinity DataKi:  14nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha3 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2(Rattus norvegicus (Rat))
Lund University

Curated by ChEMBL
LigandPNGBDBM50293262(2-(5-benzyl-2-hydroxyphenyl)-6-methylquinolin-4(1H...)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha2beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9Q3ZPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-2(Rattus norvegicus (Rat))
Lund University

Curated by ChEMBL
LigandPNGBDBM50293263(2-(5-benzyl-2-hydroxyphenyl)-6-methyl-4H-chromen-4...)copy SMILEScopy InChI
Affinity DataKi:  19nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha2beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9Q3ZPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50185293(6-bromo-3-ethoxycarbonyl-4-quinolone | CHEMBL20525...)copy SMILEScopy InChI
Affinity DataKi:  26nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha3 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MZ2PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(RAT)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293262(2-(5-benzyl-2-hydroxyphenyl)-6-methylquinolin-4(1H...)copy SMILEScopy InChI
Affinity DataKi:  31nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha3beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9Q3ZPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))
Lund University

Curated by ChEMBL
LigandPNGBDBM50293264(2-(5-bromo-2-hydroxyphenyl)-6-methylquinolin-4(1H)...)copy SMILEScopy InChI
Affinity DataKi:  39nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha1beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9Q3ZPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM26266(Ambien | CHEMBL911 | Dalparan | N,N-dimethyl-2-[6-...)copy SMILEScopy InChI
Affinity DataKi:  53nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha1 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333161(2-(4-Methylphenyl)-9-(2-phenylethyl)-2,6-dihydro[1...)copy SMILEScopy InChI
Affinity DataKi:  65nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha2beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038FKPubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333161(2-(4-Methylphenyl)-9-(2-phenylethyl)-2,6-dihydro[1...)copy SMILEScopy InChI
Affinity DataKi:  66nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha5beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z038FKPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50185296(6-ethyl-3-(3-methylbutoxycarbonyl)-4-quinolone | C...)copy SMILEScopy InChI
Affinity DataKi:  89nMAssay Description:Displacement of [3H]Flumazenil from human GABA-Aalpha3 receptor plus beta-2-gamma-2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MZ2PubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3(RAT)
Lund University

Curated by ChEMBL
LigandPNGBDBM50293264(2-(5-bromo-2-hydroxyphenyl)-6-methylquinolin-4(1H)...)copy SMILEScopy InChI
Affinity DataKi:  99nMAssay Description:Displacement of [3H]flumazenil in rat GABAAalpha3beta3gamma2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9Q3ZPubMed
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